SCHEMBL19202591

SCHEMBL19202591

COC(=O)c1ccnc(N2CC(O)(c3ccc(O)cc3Cl)C2)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 5/20 0.45
HSD17B13 Q7Z5P4 1/20 0.45
KDM5A P29375 5/20 0.43
KDM5B Q9UGL1 5/20 0.43
HRH3 Q9Y5N1 2/20 0.41
PIK3CA P42336 1/20 0.39
KDM4C Q9H3R0 2/20 0.39
KDM4E B2RXH2 2/20 0.38
KDM6B O15054 1/20 0.38
KDM5C P41229 1/20 0.38
KDM2A Q9Y2K7 1/20 0.38
KDM3A Q9Y4C1 1/20 0.38
ACLY P53396 1/20 0.38
JMJD6 Q6NYC1 1/20 0.37
ALOX15 P16050 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 1/20 0.36
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17843286 0.90 HRH3 (0.43) NR1H4HSD17B13KDM5AKDM5BHRH3
SCHEMBL29139868 0.88 NR1H4 (0.44) NR1H4HSD17B13KDM5AKDM5BPIK3CA
SCHEMBL30775159 0.87 NR1H4 (0.53) NR1H4HSD17B13KDM5AKDM5BPIK3CA
SCHEMBL29139872 0.87 NR1H4 (0.53) NR1H4HSD17B13KDM5AKDM5BPIK3CA
Nitrous Acid SCHEMBL29139870 0.83 NR1H4 (0.51) NR1H4HSD17B13KDM5AKDM5BPIK3CA
SCHEMBL19202590 0.83 NR1H4 (0.46) NR1H4HSD17B13KDM5AKDM5BHRH3
SCHEMBL19689507 0.78 NR1H4 (0.51) NR1H4
SCHEMBL30775162 0.78 NR1H4 (0.51) NR1H4
SCHEMBL17843228 0.78 CRBN (0.52) NR1H4HRH3
SCHEMBL19689487 0.76 MALT1 (0.40) NR1H4HSD17B13HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017128896-A1 FXR AGONIST AND PREPARATION METHOD AND USE THEREOF 江苏豪森药业集团有限公司 2017-08-03 WO disclosed