SCHEMBL30780259

SCHEMBL30780259

CCC(=O)c1cc(C)c(-c2cc3cnc(N)cc3n3ncnc23)cn1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 2/20 0.32
GABRD O14764 2/20 0.32
GABRA1 P14867 2/20 0.32
GABRB1 P18505 2/20 0.32
GABRG2 P18507 2/20 0.32
GABRB3 P28472 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRA3 P34903 2/20 0.32
GABRA2 P47869 2/20 0.32
GABRB2 P47870 2/20 0.32
GABRA4 P48169 2/20 0.32
GABRE P78334 2/20 0.32
GABRA6 Q16445 2/20 0.32
GABRG1 Q8N1C3 2/20 0.32
GABRG3 Q99928 2/20 0.32
GABRQ Q9UN88 2/20 0.32
ABL1 P00519 1/20 0.32
KDM4E B2RXH2 2/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27142827 1.00 GABRP (0.32) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL30780162 0.88 ABL1 (0.32) GABRG2GABRB3GABRA5ABL1NPC1
SCHEMBL27137472 0.88 ABL1 (0.32) GABRG2GABRB3GABRA5ABL1NPC1
SCHEMBL30780121 0.82 ABL1 (0.39) ABL1
SCHEMBL27145391 0.82 ABL1 (0.39) ABL1
SCHEMBL30780126 0.82 ABL1 (0.36) ABL1FGFR1SRCPIK3R1PIK3CA
SCHEMBL27135758 0.82 ABL1 (0.36) ABL1FGFR1SRCPIK3R1PIK3CA
SCHEMBL27142787 0.82 ABL1 (0.36) ABL1FGFR1SRCPIK3R1PIK3CA
SCHEMBL30780272 0.82 GABRP (0.32) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL27152884 0.82 GABRP (0.32) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4577546-A1 NAPHTHYRIDINE COMPOUNDS FOR INHIBITION OF RAF KINASES Enliven Inc. (US) 2025-07-02 EP disclosed
CN-120129682-A Naphthyridine compounds for inhibition of RAF kinase 英莱汶公司 2025-06-10 CN disclosed
WO-2024044713-A1 NAPHTHYRIDINE COMPOUNDS FOR INHIBITION OF RAF KINASES ENLIVEN INC. (US) 2024-02-29 WO disclosed