SCHEMBL30780288

SCHEMBL30780288

CC(C)(C)OC(=O)Nc1cc2c(cn1)cc(Cl)n1ccnc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.44
DYRK1A Q13627 1/20 0.44
ATR Q13535 1/20 0.36
BRD4 O60885 1/20 0.36
MAPKAPK2 P49137 2/20 0.35
RORC P51449 1/20 0.35
TSHR P16473 1/20 0.35
FSHR P23945 1/20 0.35
CDK9 P50750 2/20 0.35
IRAK4 Q9NWZ3 1/20 0.34
TLR9 Q9NR96 1/20 0.34
TLR8 Q9NR97 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
PTGER1 P34995 2/20 0.33
MAPK1 P28482 1/20 0.33
P2RX3 P56373 1/20 0.33
CYP2C9 P11712 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2B P29275 1/20 0.33
ABL1 P00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27138078 0.84 GSK3B (0.45) GSK3BDYRK1AATRBRD4MAPKAPK2
SCHEMBL27152501 0.83 ABL1 (0.35) GSK3BDYRK1AABL1
SCHEMBL30780156 0.76 GSK3B (0.36) GSK3BDYRK1ABRD4TLR9TLR8
SCHEMBL10288086 0.73 GSK3B (0.54) GSK3BDYRK1AATRMAPKAPK2CDK9
SCHEMBL18308988 0.70 GSK3B (0.47) GSK3BDYRK1AATRMAPKAPK2RORC
SCHEMBL21287636 0.70 BRD4 (0.35) GSK3BDYRK1AATRBRD4IRAK4
SCHEMBL20520009 0.69 GSK3B (0.47) GSK3BDYRK1AATRMAPKAPK2RORC
SCHEMBL14151806 0.69 GSK3B (0.55) GSK3BDYRK1AMAPKAPK2CDK9IRAK4
SCHEMBL30636341 0.68 GSK3B (0.60) GSK3BDYRK1AMAPK1ABL1
SCHEMBL28166698 0.68 GSK3B (0.60) GSK3BDYRK1AMAPK1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4577546-A1 NAPHTHYRIDINE COMPOUNDS FOR INHIBITION OF RAF KINASES Enliven Inc. (US) 2025-07-02 EP disclosed
WO-2024044713-A1 NAPHTHYRIDINE COMPOUNDS FOR INHIBITION OF RAF KINASES ENLIVEN INC. (US) 2024-02-29 WO disclosed