SCHEMBL30788998

SCHEMBL30788998

FC(F)(F)c1ccc(-c2ccc(-c3nc4ccc(Cl)cc4o3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 2/20 0.51
SMN1; SMN2 Q16637 3/20 0.50
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
HPGD P15428 2/20 0.50
LMNA P02545 1/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
TLR9 Q9NR96 1/20 0.50
PIK3CG P48736 1/20 0.50
HDAC6 Q9UBN7 2/20 0.49
HDAC3 O15379 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
CASP3 P42574 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
ESR1 P03372 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18935939 0.86 TLR9 (0.55) SMN1; SMN2KDM4EALDH1A1HPGDTLR9
SCHEMBL10590678 0.85 SMN1; SMN2 (0.61) SMN1; SMN2KDM4EALDH1A1HPGDLMNA
SCHEMBL23748384 0.84 HDAC6 (0.56) CETPSMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL30789017 0.84 HDAC6 (0.56) CETPSMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL25026542 0.83 HDAC3 (0.60) CETPSMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL23748387 0.82 SMN1; SMN2 (0.71) SMN1; SMN2KDM4EALDH1A1HPGDLMNA
SCHEMBL2245453 0.81 NPC1 (0.67) SMN1; SMN2KDM4EALDH1A1HPGDLMNA
SCHEMBL17199136 0.81 NPC1 (0.74) SMN1; SMN2KDM4EALDH1A1HPGDNFKB1
SCHEMBL14243239 0.81 HDAC6 (0.53) SMN1; SMN2KDM4EALDH1A1HPGDTLR9
SCHEMBL8740136 0.81 ESR1 (0.74) TLR9HDAC6HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113195084-B Benzoxazoles and related compounds useful as modulators of chaperone mediated autophagy 阿尔伯爱因斯坦医学院 2024-04-09 CN claimed
CN-113195084-B Benzoxazoles and related compounds useful as modulators of chaperone mediated autophagy 阿尔伯爱因斯坦医学院 2024-04-09 CN disclosed