SCHEMBL30794812

SCHEMBL30794812

Cc1c(C(=O)NCc2cccc(F)c2)c(=S)n(C)c2cc(C(F)(F)F)ccc12

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.48
CCR1 P32246 7/20 0.45
MLYCD O95822 1/20 0.43
S1PR3 Q99500 2/20 0.43
GLS O94925 1/20 0.43
MAPT P10636 1/20 0.42
MEN1 O00255 1/20 0.41
PLA2G1B P04054 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41
MAPK14 Q16539 1/20 0.40
KIF11 P52732 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28973 1.00 ROCK2 (0.48) ROCK2CCR1MLYCDS1PR3GLS
SCHEMBL30795780 0.90 ROCK2 (0.48) ROCK2CCR1MLYCDS1PR3GLS
SCHEMBL715292 0.90 ROCK2 (0.48) ROCK2CCR1MLYCDS1PR3GLS
SCHEMBL30796474 0.89 MEN1 (0.46) CCR1S1PR3MAPTMEN1GAA
SCHEMBL29573 0.89 MEN1 (0.46) CCR1S1PR3MAPTMEN1GAA
SCHEMBL30795738 0.83 S1PR3 (0.47) ROCK2CCR1MLYCDS1PR3GLS
SCHEMBL30795875 0.83 S1PR3 (0.45) ROCK2CCR1MLYCDS1PR3GLS
SCHEMBL715295 0.83 S1PR3 (0.47) ROCK2CCR1MLYCDS1PR3GLS
SCHEMBL29002 0.83 S1PR3 (0.45) ROCK2CCR1MLYCDS1PR3GLS
SCHEMBL716049 0.82 S1PR3 (0.50) CCR1MLYCDS1PR3MAPTMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4584250-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS Biohaven Therapeutics Ltd. (VG) 2025-07-16 EP disclosed
EP-4580679-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS AND NMDA RECEPTOR ANTAGONISTS Biohaven Therapeutics Ltd. (VG) 2025-07-09 EP disclosed
WO-2024054811-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-14 WO disclosed
WO-2024054807-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS AND TDP-43 MODULATORS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-14 WO disclosed
WO-2024050389-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS AND NMDA RECEPTOR ANTAGONISTS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-07 WO disclosed