Dideazafolate

Dideazafolate

SCHEMBL30799321

Nc1nc2ccc(CNc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)cc2c(=O)[nH]1

nearest known ligand 0.90

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DHFR P00374 10/20 0.90
ATIC P31939 2/20 0.72
TYMS P04818 2/20 0.72
GART P22102 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dideazafolate SCHEMBL10036542 1.00 DHFR (0.90) DHFRATICTYMSGART
SCHEMBL29692260 0.95 DHFR (1.00) DHFRATICTYMSGART
SCHEMBL6449047 0.92 DHFR (0.77) DHFRATICTYMSGART
SCHEMBL24413576 0.91 DHFR (0.76) DHFRATICTYMSGART
SCHEMBL24413587 0.91 DHFR (0.76) DHFRATICTYMSGART
SCHEMBL410474 0.91 DHFR (0.76) DHFRATICTYMSGART
SCHEMBL15507841 0.91 DHFR (0.75) DHFRATICTYMSGART
SCHEMBL29617327 0.90 DHFR (0.74) DHFRATICTYMSGART
SCHEMBL408871 0.89 DHFR (0.72) DHFRATICTYMSGART
Dideazafolate SCHEMBL13125706 0.88 DHFR (0.70) DHFRATICTYMSGART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111989138-B Humanized anti-Prostate Specific Membrane Antigen (PSMA) antibody drug conjugates AMBRX公司 2024-02-09 CN disclosed
CN-117440833-A anti-HER 2 antibody-drug conjugates and uses thereof AMBRX公司 2024-01-23 CN disclosed