SCHEMBL30801141

SCHEMBL30801141

COC(=O)N1Cc2cccc(Br)c2C[C@@H]1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.43
POLB P06746 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
AGTR2 P50052 1/20 0.41
ABHD6 Q9BV23 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16267600 1.00 ACE (0.43) ACEPOLBTDP1AGTR2ABHD6
SCHEMBL16271276 0.90 CYP19A1 (0.41) AGTR2ABHD6
SCHEMBL31652041 0.90 CYP19A1 (0.41) AGTR2ABHD6
SCHEMBL9849174 0.90 CYP19A1 (0.41) AGTR2ABHD6
SCHEMBL29570670 0.90 CYP19A1 (0.41) AGTR2ABHD6
SCHEMBL16267710 0.85 POLB (0.43) ACEPOLBTDP1AGTR2ABHD6
SCHEMBL9849125 0.85 POLB (0.43) ACEPOLBTDP1AGTR2ABHD6
SCHEMBL32676636 0.81 CYP19A1 (0.45) AGTR2ABHD6
SCHEMBL20483181 0.81 PTPN1 (0.53) ABHD6
SCHEMBL32676746 0.81 CYP19A1 (0.45) AGTR2ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111971282-B Pyrazolotetrahydroisoquinoline derivatives as dopamine D1 receptor positive modulators 伊莱利利公司 2024-03-19 CN disclosed