SCHEMBL30801448

SCHEMBL30801448

COCOc1cc(-c2ccc3c(N4CC5CCC(C4)N5C(=O)OC(C)(C)C)nc(OCC=O)nc3c2F)c2c(C#C[Si](C(C)C)(C(C)C)C(C)C)c(F)ccc2c1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 3/20 0.33
JAK2 O60674 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
KRAS P01116 4/20 0.32
GPR119 Q8TDV5 3/20 0.32
MAPK3 P27361 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30131075 1.00 JAK1 (0.33) JAK1JAK2TYK2JAK3KRAS
SCHEMBL31129339 0.94 KRAS (0.39) KRASMAPK3MAPK1
SCHEMBL31129721 0.94 KRAS (0.39) KRASMAPK3MAPK1
SCHEMBL31129533 0.94 KRAS (0.39) KRASMAPK3MAPK1
SCHEMBL30131061 0.93 JAK1 (0.33) JAK1JAK2TYK2JAK3KRAS
SCHEMBL30801453 0.93 JAK1 (0.33) JAK1JAK2TYK2JAK3KRAS
SCHEMBL30864096 0.92 KRAS (0.34) JAK1JAK2TYK2JAK3KRAS
SCHEMBL30782214 0.91 JAK1 (0.35) JAK1JAK2TYK2JAK3GPR119
SCHEMBL30779081 0.91 JAK1 (0.35) JAK1JAK2TYK2JAK3GPR119
SCHEMBL30864064 0.91 KRAS (0.34) JAK1JAK2TYK2JAK3KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117460737-A Heteroaromatic compounds, method for the production and use thereof 四川科伦博泰生物医药股份有限公司 2024-01-26 CN disclosed