SCHEMBL30808641

SCHEMBL30808641

O=C(O)CN1C(=O)CSc2cc(C(F)(F)F)ccc21

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
PKM P14618 1/20 0.47
MEN1 O00255 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
KMT2A Q03164 1/20 0.46
FPR2 P25090 1/20 0.45
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
NPSR1 Q6W5P4 2/20 0.43
HSD17B3 P37058 1/20 0.41
GAA P10253 2/20 0.40
ALOX15 P16050 1/20 0.39
SLC5A1 P13866 2/20 0.39
SLC5A2 P31639 2/20 0.39
RAD52 P43351 1/20 0.39
HPGD P15428 1/20 0.38
KCNN4 O15554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10511510 0.91 ALDH1A1 (0.56) ALDH1A1PKMMEN1GSK3AGSK3B
SCHEMBL30808658 0.87 ALDH1A1 (0.46) ALDH1A1PKMMEN1KMT2AFPR2
SCHEMBL10648891 0.84 TSHR (0.48) ALDH1A1MEN1GSK3AGSK3BKMT2A
SCHEMBL4328088 0.81 NPY5R (0.51) MEN1GSK3AGSK3BKMT2ANPSR1
SCHEMBL10511901 0.79 KCNN4 (0.46) ALDH1A1PKMMEN1GSK3AGSK3B
SCHEMBL29456205 0.78 NOTUM (0.50) ALDH1A1MEN1KMT2AFPR2TP53
SCHEMBL3782479 0.78 NOTUM (0.50) ALDH1A1MEN1KMT2AFPR2TP53
SCHEMBL30808603 0.78 MEN1 (0.50) ALDH1A1MEN1GSK3AGSK3BKMT2A
SCHEMBL4971618 0.77 NPSR1 (0.67) ALDH1A1MEN1GSK3AGSK3BKMT2A
SCHEMBL30808619 0.77 NPSR1 (0.67) ALDH1A1MEN1GSK3AGSK3BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023250002-A1 IDENTIFICATION OF NOVEL BENZOTHIAZONES AS TAU-SH3 INTERACTION INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE SOUTHERN RESEARCH INSTITUTE (US) 2023-12-28 WO disclosed