SCHEMBL30822689

SCHEMBL30822689

Cc1cc(-n2c([C@H](C)N)cc3cccc(C)c3c2=O)n[nH]1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
PIK3R1 P27986 3/20 0.38
PIK3CA P42336 2/20 0.38
PIK3CD O00329 8/20 0.37
PIK3CG P48736 3/20 0.37
MAPK1 P28482 1/20 0.33
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32
GFER P55789 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
JAK1 P23458 2/20 0.32
TYK2 P29597 2/20 0.32
JAK3 P52333 2/20 0.32
JAK2 O60674 1/20 0.32
PIK3R2 O00459 1/20 0.31
AURKA O14965 1/20 0.31
AURKB Q96GD4 1/20 0.31
ABCB11 O95342 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29164574 1.00 CYP1A2 (0.38) CYP1A2PIK3R1PIK3CAPIK3CDPIK3CG
SCHEMBL29164573 1.00 CYP1A2 (0.38) CYP1A2PIK3R1PIK3CAPIK3CDPIK3CG
SCHEMBL30822713 0.89 PIK3R1 (0.41) CYP1A2PIK3R1PIK3CAPIK3CDPIK3CG
SCHEMBL29164722 0.89 PIK3R1 (0.41) CYP1A2PIK3R1PIK3CAPIK3CDPIK3CG
SCHEMBL29164724 0.89 PIK3R1 (0.41) CYP1A2PIK3R1PIK3CAPIK3CDPIK3CG
SCHEMBL30822729 0.89 PIK3CD (0.40) PIK3R1PIK3CAPIK3CDPIK3CGPIK3R2
SCHEMBL29164738 0.89 PIK3CD (0.37) PIK3R1PIK3CAPIK3CDPIK3CGMAPK1
SCHEMBL29164734 0.89 PIK3CD (0.37) PIK3R1PIK3CAPIK3CDPIK3CGMAPK1
SCHEMBL29164550 0.89 PIK3CD (0.40) PIK3R1PIK3CAPIK3CDPIK3CGPIK3R2
SCHEMBL30822691 0.89 PIK3CD (0.37) PIK3R1PIK3CAPIK3CDPIK3CGMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117659001-A Aminopyrimidine derivatives and their use in medicine 广东东阳光药业股份有限公司 2024-03-08 CN disclosed