SCHEMBL30822720

SCHEMBL30822720

Cc1cc(-n2ccc3ccc(F)cc3c2=O)n[nH]1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 7/20 0.49
SYK P43405 3/20 0.41
NTRK1 P04629 9/20 0.40
TYMS P04818 2/20 0.39
AURKA O14965 3/20 0.38
JAK2 O60674 1/20 0.36
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
CASP3 P42574 1/20 0.35
AURKB Q96GD4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30822704 0.86 ALK (0.36) ALKTYMS
SCHEMBL30822718 0.84 TYMS (0.39) ALKSYKTYMSAURKA
SCHEMBL30822708 0.82 AURKA (0.41) ALKSYKAURKAAURKB
SCHEMBL30822734 0.78 TYMS (0.35) TYMS
SCHEMBL30822741 0.75 ALK (0.41) ALKNTRK1AURKAJAK2AURKB
SCHEMBL29164558 0.73 SYK (0.41) ALKSYKNTRK1JAK2CASP3
SCHEMBL29164556 0.73 SYK (0.41) ALKSYKNTRK1JAK2CASP3
SCHEMBL30822680 0.73 SYK (0.41) ALKSYKNTRK1JAK2CASP3
SCHEMBL30822710 0.72 CYP1A2 (0.40) ALKAURKAJAK2AURKB
SCHEMBL30822709 0.71 ALK (0.36) ALKSYKNTRK1AURKAJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117659001-A Aminopyrimidine derivatives and their use in medicine 广东东阳光药业股份有限公司 2024-03-08 CN disclosed