SCHEMBL30824751

SCHEMBL30824751

O=C(CCC(=O)N1CCc2ccccc2C1c1ccccc1)NCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HHAT Q5VTY9 3/20 0.56
CYP2D6 P10635 1/20 0.55
HDAC8 Q9BY41 4/20 0.52
HDAC3 O15379 3/20 0.52
HDAC1 Q13547 3/20 0.52
HDAC2 Q92769 3/20 0.52
NCOR2 Q9Y618 3/20 0.52
CHRM3 P20309 4/20 0.48
CHRM2 P08172 2/20 0.48
CHRM1 P11229 2/20 0.48
CACNA1F O60840 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
KCNE1 P15382 1/20 0.47
KCNQ1 P51787 1/20 0.47
CACNA1D Q01668 1/20 0.47
KCNH2 Q12809 1/20 0.47
CACNA1S Q13698 1/20 0.47
CACNA1C Q13936 1/20 0.47
SCN5A Q14524 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3240992 1.00 HHAT (0.56) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL3242938 0.93 CHRM3 (0.55) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL30795961 0.93 HHAT (0.54) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL30795434 0.93 HHAT (0.52) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL30795853 0.93 CHRM3 (0.55) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL3236277 0.93 HHAT (0.52) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL3232980 0.93 HHAT (0.54) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL3236487 0.90 HDAC8 (0.54) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL3235146 0.90 CHRM3 (0.52) HHATCYP2D6HDAC8HDAC3HDAC1
SCHEMBL3235270 0.90 TRPM8 (0.56) HHATCYP2D6HDAC8HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024054807-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS AND TDP-43 MODULATORS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-14 WO disclosed