SCHEMBL30824934

SCHEMBL30824934

Cc1cc([N+](=O)[O-])ccc1C(=O)N1CCCCc2cc(Cl)ccc21

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 7/20 0.70
AVPR1A P37288 3/20 0.52
LMNA P02545 3/20 0.50
NPC1 O15118 1/20 0.50
MAPT P10636 1/20 0.50
HTT P42858 1/20 0.50
HDAC1 Q13547 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
DRD4 P21917 1/20 0.48
ALDH1A1 P00352 1/20 0.47
RECQL P46063 1/20 0.47
RAB9A P51151 1/20 0.47
PAX8 Q06710 1/20 0.47
NOTUM Q6P988 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1291539 0.84 AVPR2 (0.50) AVPR2AVPR1ALMNANPC1MAPT
SCHEMBL30824950 0.84 AVPR2 (0.50) AVPR2AVPR1ALMNANPC1MAPT
SCHEMBL30354667 0.83 AVPR2 (0.76) AVPR2AVPR1AHDAC1HDAC6NOTUM
SCHEMBL26406287 0.81 AVPR2 (0.46) AVPR2AVPR1ALMNANPC1MAPT
SCHEMBL28475504 0.79 AVPR2 (0.49) AVPR2AVPR1ALMNANPC1HTT
SCHEMBL8671412 0.78 AVPR2 (0.67) AVPR2LMNANPC1MAPTHTT
SCHEMBL4680537 0.77 AVPR2 (0.47) AVPR2AVPR1ALMNANPC1HTT
SCHEMBL7355229 0.77 AVPR2 (0.52) AVPR2LMNANPC1MAPTHTT
SCHEMBL7245901 0.77 AVPR2 (0.73) AVPR2AVPR1ALMNAHDAC1HDAC6
SCHEMBL5486199 0.77 AVPR2 (0.47) AVPR2AVPR1ALMNANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117624049-A Method for synthesizing and refining key intermediate of tolvaptan 山东科新药业有限公司 2024-03-01 CN claimed
CN-117624049-A Method for synthesizing and refining key intermediate of tolvaptan 山东科新药业有限公司 2024-03-01 CN disclosed