SCHEMBL30833642

SCHEMBL30833642

CN(c1ccccc1Nc1nc(Nc2ccc3cnn(C)c3c2)ncc1Cl)S(C)(=O)=O

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 9/20 0.63
MET P08581 3/20 0.63
EGFR P00533 3/20 0.51
AXL P30530 6/20 0.49
AURKA O14965 1/20 0.47
AURKB Q96GD4 1/20 0.47
NEK2 P51955 1/20 0.47
INSR P06213 3/20 0.47
PTK2 Q05397 2/20 0.47
FLT3 P36888 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190681 1.00 ALK (0.63) ALKMETEGFRAXLAURKA
SCHEMBL30833727 0.81 ALK (0.47) ALKMETEGFRAXLAURKA
SCHEMBL30429763 0.81 CDK2 (0.47) ALKEGFRAXL
SCHEMBL29833077 0.80 EGFR (0.62) ALKEGFRINSRPTK2
SCHEMBL28996874 0.80 EGFR (0.62) ALKEGFRINSRPTK2
SCHEMBL21432463 0.80 AXL (0.73) ALKMETEGFRAXLAURKA
SCHEMBL25233510 0.79 AURKA (0.67) ALKMETEGFRAXLAURKA
SCHEMBL21432456 0.78 EGFR (0.71) ALKMETEGFRAXLNEK2
SCHEMBL25284886 0.78 ALK (0.65) ALKMETEGFRAURKAAURKB
SCHEMBL29190658 0.78 ALK (0.59) ALKMETEGFRFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed