SCHEMBL30833727

SCHEMBL30833727

CNS(=O)(=O)Cc1ccccc1Nc1nc(Nc2ccc3cnn(C)c3c2)ncc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 7/20 0.47
INSR P06213 3/20 0.47
MET P08581 4/20 0.46
CDK9 P50750 3/20 0.45
AURKA O14965 2/20 0.45
NEK2 P51955 2/20 0.45
CDC7 O00311 2/20 0.45
JAK2 O60674 2/20 0.45
ROCK2 O75116 2/20 0.45
PRKD3 O94806 2/20 0.45
MAP4K4 O95819 2/20 0.45
PAK4 O96013 2/20 0.45
PRKACA P17612 2/20 0.45
CLK2 P49760 2/20 0.45
GSK3A P49840 2/20 0.45
CDK7 P50613 2/20 0.45
PRKX P51817 2/20 0.45
CAMK2D Q13557 2/20 0.45
DYRK1A Q13627 2/20 0.45
MELK Q14680 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833714 0.84 ALK (0.46) ALKINSRMETCDK9AURKA
SCHEMBL30833642 0.81 ALK (0.63) ALKINSRMETAURKANEK2
SCHEMBL29190681 0.81 ALK (0.63) ALKINSRMETAURKANEK2
SCHEMBL30429763 0.81 CDK2 (0.47) ALKCDK9CDC7JAK2ROCK2
SCHEMBL28996874 0.80 EGFR (0.62) ALKINSRPTK2EGFRIGF1R
SCHEMBL29833077 0.80 EGFR (0.62) ALKINSRPTK2EGFRIGF1R
SCHEMBL30833783 0.78 SYK (0.47) ALKMETCDK9CDC7JAK2
SCHEMBL30833667 0.78 KDR (0.48) CDK9CDC7JAK2ROCK2MAP4K4
SCHEMBL29190658 0.76 ALK (0.59) ALKMETFLT3EGFRROS1
SCHEMBL31251206 0.73 EGFR (0.63) ALKINSRPTK2EGFRIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed