SCHEMBL30833646

SCHEMBL30833646

CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc3cnn(C)c3c2)ncc1Br

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 15/20 0.55
CDK7 P50613 1/20 0.54
CDK9 P50750 1/20 0.54
MET P08581 10/20 0.50
PTK2 Q05397 3/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
ULK1 O75385 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190577 1.00 ALK (0.55) ALKCDK7CDK9METPTK2
SCHEMBL31251238 0.93 ALK (0.55) ALKCDK7CDK9METPTK2
SCHEMBL29190525 0.90 ALK (0.68) ALKCDK7CDK9PTK2ULK1
SCHEMBL30833701 0.90 ALK (0.68) ALKCDK7CDK9PTK2ULK1
SCHEMBL31251116 0.86 ALK (0.56) ALKCDK7CDK9METPTK2
SCHEMBL31251128 0.86 CDK7 (0.54) ALKCDK7CDK9METPTK2
SCHEMBL32690407 0.83 CDK7 (0.54) ALKCDK7CDK9METPTK2
SCHEMBL31251329 0.83 ALK (0.68) ALKCDK7CDK9ULK1
SCHEMBL30833810 0.82 ALK (0.49) ALKCDK7CDK9
SCHEMBL29190704 0.82 ALK (0.49) ALKCDK7CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed