SCHEMBL30833701

SCHEMBL30833701

Cn1ncc2ccc(Nc3ncc(Br)c(Nc4ccccc4S(C)(=O)=O)n3)cc21

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 6/20 0.68
ULK1 O75385 1/20 0.50
CDK2 P24941 2/20 0.48
CDK1 P06493 1/20 0.48
KDR P35968 1/20 0.48
ZAP70 P43403 6/20 0.47
CDK19 Q9BWU1 3/20 0.47
CDC7 O00311 1/20 0.46
DAPK3 O43293 1/20 0.46
JAK2 O60674 1/20 0.46
ROCK2 O75116 1/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
PAK4 O96013 1/20 0.46
PIM1 P11309 1/20 0.46
PRKACA P17612 1/20 0.46
SYK P43405 1/20 0.46
CSNK1A1 P48729 1/20 0.46
CDK8 P49336 1/20 0.46
CLK2 P49760 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190525 1.00 ALK (0.68) ALKULK1CDK2CDK1KDR
SCHEMBL31251329 0.93 ALK (0.68) ALKULK1CDK2CDK1KDR
SCHEMBL29190577 0.90 ALK (0.55) ALKULK1CDK7CDK9PTK2
SCHEMBL30833646 0.90 ALK (0.55) ALKULK1CDK7CDK9PTK2
SCHEMBL29190704 0.85 ALK (0.49) ALKCDK2CDK1KDRCDK19
SCHEMBL30833810 0.85 ALK (0.49) ALKCDK2CDK1KDRCDK19
SCHEMBL31251169 0.84 ALK (0.62) ALKULK1CDK2CDK1KDR
SCHEMBL31251390 0.84 ALK (0.65) ALKULK1CDK2CDK1KDR
SCHEMBL29190613 0.83 ALK (0.49) ALKCDK2CDK19CDC7DAPK3
SCHEMBL30833747 0.83 ALK (0.49) ALKCDK2CDK19CDC7DAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed