SCHEMBL30833746

SCHEMBL30833746

CNS(=O)(=O)Cc1ccccc1Nc1nc(Nc2ccc3cn[nH]c3c2)ncc1Br

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.51
FGFR1 P11362 2/20 0.51
ZAP70 P43403 3/20 0.50
ULK1 O75385 1/20 0.45
SYK P43405 7/20 0.45
CDK2 P24941 3/20 0.45
DAPK3 O43293 2/20 0.45
PRKD3 O94806 2/20 0.45
MAP4K4 O95819 2/20 0.45
PAK4 O96013 2/20 0.45
PIM1 P11309 2/20 0.45
PRKACA P17612 2/20 0.45
FLT3 P36888 2/20 0.45
CSNK1A1 P48729 2/20 0.45
CLK2 P49760 2/20 0.45
CDK9 P50750 2/20 0.45
JAK3 P52333 2/20 0.45
CDK5 Q00535 2/20 0.45
MAP4K2 Q12851 2/20 0.45
STK3 Q13188 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190561 0.80 EGFR (0.52) EGFRFGFR1ZAP70SYKCDK2
SCHEMBL30833756 0.79 EGFR (0.57) EGFRFGFR1ZAP70SYKCDK2
SCHEMBL29190600 0.79 EGFR (0.57) EGFRFGFR1ZAP70SYKCDK2
SCHEMBL30833657 0.78 ZAP70 (0.43) EGFRFGFR1ZAP70ULK1SYK
SCHEMBL29190651 0.78 EGFR (0.54) EGFRFGFR1ZAP70SYKCDK2
SCHEMBL30833624 0.78 EGFR (0.54) EGFRFGFR1ZAP70SYKCDK2
SCHEMBL29190543 0.77 EGFR (0.51) EGFRFGFR1ZAP70SYKCDK2
SCHEMBL30833764 0.74 IGF1R (0.45) EGFRFGFR1ULK1SYKCDK2
SCHEMBL30833738 0.74 ALK (0.63) EGFRFGFR1ZAP70ULK1PRKD3
SCHEMBL6210042 0.72 PTK2 (0.55) EGFRFGFR1ULK1SYKDAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed