SCHEMBL30833802

SCHEMBL30833802

Nc1ccccc1Nc1nc(Cl)ncc1Br

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 5/20 0.55
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
EGFR P00533 3/20 0.46
CDK19 Q9BWU1 1/20 0.43
ALK Q9UM73 1/20 0.43
GAA P10253 2/20 0.41
MAPK8 P45983 2/20 0.41
PIM1 P11309 1/20 0.40
KDM1A O60341 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
LRRK2 Q5S007 1/20 0.39
MAPK10 P53779 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24260666 1.00 IGF1R (0.55) IGF1RMEN1KMT2AEGFRCDK19
SCHEMBL30833632 0.84 BCL6 (0.50) MEN1KMT2AEGFRALKGAA
SCHEMBL3340093 0.84 BCL6 (0.50) MEN1KMT2AEGFRALKGAA
SCHEMBL30833629 0.82 EGFR (0.42) IGF1RMEN1KMT2AEGFRGAA
SCHEMBL29549370 0.82 EGFR (0.42) IGF1RMEN1KMT2AEGFRGAA
SCHEMBL30833794 0.82 GAA (0.42) MEN1KMT2AEGFRGAAKDM1A
SCHEMBL600580 0.82 KMT2A (0.51) IGF1RMEN1KMT2AEGFRALK
SCHEMBL22828247 0.82 GAA (0.42) MEN1KMT2AEGFRGAAKDM1A
SCHEMBL22807434 0.82 EGFR (0.42) IGF1RMEN1KMT2AEGFRGAA
SCHEMBL17544687 0.82 IGF1R (0.55) IGF1RMEN1KMT2ACDK19ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed