SCHEMBL30834341

SCHEMBL30834341

Cc1ncc(-c2cncn2C)nc1C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.40
HTR1A P08908 2/20 0.38
HTR7 P34969 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
DRD2 P14416 1/20 0.38
HTR6 P50406 1/20 0.38
IDO1 P14902 1/20 0.35
PDPK1 O15530 1/20 0.34
GSK3B P49841 8/20 0.34
DYRK1A Q13627 8/20 0.34
LDLR P01130 1/20 0.34
PCSK9 Q8NBP7 1/20 0.34
MMP2 P08253 1/20 0.34
MMP13 P45452 1/20 0.34
MMP14 P50281 1/20 0.34
WNT1 P04628 2/20 0.33
HPGDS O60760 1/20 0.33
TGFBR1 P36897 1/20 0.33
PLK1 P53350 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25136322 0.87 LDLR (0.38) IDO1PDPK1GSK3BDYRK1ALDLR
Hydrochloric Acid SCHEMBL29182214 0.86 LDLR (0.37) IDO1PDPK1GSK3BDYRK1ALDLR
SCHEMBL30182550 0.83 GPR142 (0.37) PDPK1GSK3BDYRK1AMMP2MMP13
SCHEMBL25136313 0.83 GPR142 (0.37) PDPK1GSK3BDYRK1AMMP2MMP13
SCHEMBL25136408 0.77 PDPK1 (0.39) CYP3A4IDO1PDPK1HPGDS
Hydrochloric Acid SCHEMBL29182167 0.76 PDPK1 (0.39) CYP3A4IDO1PDPK1HPGDS
SCHEMBL25136435 0.75 PDPK1 (0.43) PDPK1GSK3BDYRK1A
SCHEMBL30182839 0.75 PDPK1 (0.43) PDPK1GSK3BDYRK1A
SCHEMBL25136318 0.73 PDPK1 (0.39) CYP3A4IDO1PDPK1GSK3BDYRK1A
SCHEMBL25136179 0.72 GSK3B (0.45) CYP2D6GSK3BDYRK1AWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117813296-A CD38 modulators and methods of use thereof 赛特凯恩蒂克公司 2024-04-02 CN disclosed