SCHEMBL30853473

SCHEMBL30853473

COC(=O)c1cc2ccccc2c(=O)n1C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
HPGD P15428 2/20 0.49
NR1H2 P55055 12/20 0.40
KDM4E B2RXH2 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
BRD4 O60885 1/20 0.38
NR1H3 Q13133 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1201914 1.00 ALDH1A1 (0.49) ALDH1A1HPGDNR1H2KDM4ENPSR1
SCHEMBL30023124 0.87 NR1H2 (0.41) ALDH1A1HPGDNR1H2KDM4ECA12
SCHEMBL23956770 0.84 USP30 (0.38) NR1H2
SCHEMBL19964584 0.84 USP30 (0.40) ALDH1A1HPGDNR1H2
SCHEMBL30396372 0.84 USP30 (0.38) NR1H2
SCHEMBL18537881 0.83 NR1H2 (0.53) NR1H2CA12CA9NR1H3
SCHEMBL30023415 0.81 DTYMK (0.41) ALDH1A1HPGDNR1H2KDM4E
SCHEMBL23930164 0.81 DTYMK (0.41) ALDH1A1HPGDNR1H2KDM4E
SCHEMBL29631893 0.77 NR1H2 (0.40) NR1H2CA12CA9NR1H3
SCHEMBL19013553 0.77 NR1H2 (0.40) NR1H2CA12CA9NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115397822-B CBP/EP300 inhibitors and uses thereof 南京药石科技股份有限公司 2024-04-16 CN disclosed