SCHEMBL30853535

SCHEMBL30853535

COc1ccccc1Nc1ncnc2c1ccn2-c1ccc(C(N)=O)c(NC2CCC(O)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 17/20 0.51
HSP90B1 P14625 1/20 0.47
HSP90AB1 P08238 1/20 0.43
BRAF P15056 1/20 0.42
CASP1 P29466 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30853519 0.93 HSP90AA1 (0.43) HSP90AA1HSP90B1BRAFCASP1
SCHEMBL30853542 0.88 HSP90AA1 (0.54) HSP90AA1HSP90B1HSP90AB1
SCHEMBL30853525 0.87 HSP90AA1 (0.57) HSP90AA1HSP90B1
SCHEMBL30853543 0.85 HSP90AA1 (0.49) HSP90AA1HSP90B1HSP90AB1
SCHEMBL30853528 0.85 PIP4K2A (0.42)
SCHEMBL30853534 0.85 HSP90AA1 (0.51) HSP90AA1HSP90B1
SCHEMBL30853518 0.84 HSP90AA1 (0.51) HSP90AA1HSP90B1HSP90AB1
SCHEMBL30853530 0.81 HSP90AA1 (0.49) HSP90AA1HSP90B1HSP90AB1
SCHEMBL30853526 0.80 PIP4K2A (0.46) HSP90AA1HSP90B1
SCHEMBL14177840 0.80 HSP90AA1 (0.62) HSP90AA1HSP90B1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118047781-A HSP90 inhibitor and preparation method and application thereof 广西大学 2024-05-17 CN disclosed