SCHEMBL30853530

SCHEMBL30853530

NC(=O)c1ccc(-n2ccc3c(Nc4ccc(C(F)(F)F)cc4)ncnc32)cc1NC1CCC(O)CC1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 13/20 0.49
PIP4K2A P48426 1/20 0.44
PIK3CG P48736 1/20 0.44
HSP90B1 P14625 2/20 0.44
HSP90AB1 P08238 2/20 0.44
TRAP1 Q12931 1/20 0.44
JAK2 O60674 3/20 0.40
JAK1 P23458 3/20 0.40
TYK2 P29597 2/20 0.40
JAK3 P52333 2/20 0.40
TRPV1 Q8NER1 1/20 0.40
EGFR P00533 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30853520 0.93 PIP4K2A (0.45) HSP90AA1PIP4K2APIK3CGJAK2JAK1
SCHEMBL30853542 0.90 HSP90AA1 (0.54) HSP90AA1PIP4K2APIK3CGHSP90B1HSP90AB1
SCHEMBL30853543 0.87 HSP90AA1 (0.49) HSP90AA1PIP4K2APIK3CGHSP90B1HSP90AB1
SCHEMBL30853534 0.86 HSP90AA1 (0.51) HSP90AA1PIP4K2APIK3CGHSP90B1
SCHEMBL30853531 0.85 PIP4K2A (0.47) HSP90AA1PIP4K2APIK3CGJAK3TRPV1
SCHEMBL30853518 0.84 HSP90AA1 (0.51) HSP90AA1PIP4K2APIK3CGHSP90B1HSP90AB1
SCHEMBL30853525 0.83 HSP90AA1 (0.57) HSP90AA1HSP90B1
SCHEMBL30853526 0.82 PIP4K2A (0.46) HSP90AA1PIP4K2APIK3CGHSP90B1JAK2
SCHEMBL30853535 0.81 HSP90AA1 (0.51) HSP90AA1HSP90B1HSP90AB1
SCHEMBL30853539 0.80 PIP4K2A (0.47) HSP90AA1PIP4K2APIK3CGHSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118047781-A HSP90 inhibitor and preparation method and application thereof 广西大学 2024-05-17 CN disclosed