SCHEMBL30856785

SCHEMBL30856785

CN1CCN(c2cc(Br)ccn2)C(=O)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
HRH4 Q9H3N8 3/20 0.35
HRH3 Q9Y5N1 1/20 0.35
RAD51 Q06609 1/20 0.34
HTT P42858 1/20 0.33
ACVR1 Q04771 1/20 0.33
BRD4 O60885 1/20 0.33
SPR P35270 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
ROCK1 Q13464 1/20 0.32
MAP3K14 Q99558 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24707424 1.00 SLC6A2 (0.37) SLC6A2SLC6A4HRH4HRH3RAD51
SCHEMBL30856775 0.84 GRIN2D (0.47) SLC6A2SLC6A4HRH4HRH3ACVR1
SCHEMBL24706831 0.84 GRIN2D (0.47) SLC6A2SLC6A4HRH4HRH3ACVR1
SCHEMBL901368 0.79 ALDH1A1 (0.40) KDM4EALDH1A1SMN1; SMN2ACACB
SCHEMBL13063401 0.79 CYP17A1 (0.48) HRH3KDM4EALDH1A1
SCHEMBL12835924 0.77 CRBN (0.49) KDM4EALDH1A1SMN1; SMN2
SCHEMBL24135526 0.77 PARP1 (0.48) ALDH1A1ROCK1MAP3K14CYP3A4CYP2C9
SCHEMBL31333194 0.76 PARP1 (0.47) ROCK1MAP3K14
SCHEMBL29187003 0.75 MEN1 (0.36) SLC6A2SLC6A4HRH4HRH3ACVR1
SCHEMBL15509065 0.74 HRH4 (0.59) HRH4HRH3HTTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117813302-A Substituted tetrahydrofuran-2-carboxamides as sodium channel modulators 沃泰克斯药物股份有限公司 2024-04-02 CN disclosed