SCHEMBL30857549

SCHEMBL30857549

COC(=O)c1ccc(N2CCN(CC3=C(c4ccc(Cl)cc4)CCC(C)(C)C3)C[C@@H]2CCO[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BCL2L1 Q07817 14/20 0.50
BCL2 P10415 17/20 0.46
BAD Q92934 2/20 0.38
BCL2L11 O43521 1/20 0.38
CYP2C9 P11712 1/20 0.38
MCL1 Q07820 1/20 0.38
ASPH Q12797 1/20 0.38
BCL2L2 Q92843 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30857677 0.93 BCL2L1 (0.51) BCL2L1BCL2BADBCL2L11CYP2C9
SCHEMBL30857629 0.93 BCL2L1 (0.51) BCL2L1BCL2BADBCL2L11CYP2C9
SCHEMBL30857651 0.88 BCL2L1 (0.44) BCL2L1BCL2BADBCL2L11CYP2C9
SCHEMBL30857578 0.87 BCL2L1 (0.59) BCL2L1BCL2BADBCL2L11CYP2C9
SCHEMBL30857642 0.83 KMT2A (0.45) CYP2C9
SCHEMBL21751667 0.80 BCL2L1 (0.59) BCL2L1BCL2BADBCL2L11CYP2C9
SCHEMBL30857743 0.79 BCL2L1 (0.69) BCL2L1BCL2BADBCL2L11CYP2C9
SCHEMBL30857524 0.77 BCL2L1 (0.71) BCL2L1BCL2BADBCL2L11CYP2C9
SCHEMBL23164961 0.74 BCL2L1 (0.51) BCL2L1BCL2BCL2L2
SCHEMBL21751607 0.74 BCL2L1 (0.51) BCL2L1BCL2BCL2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024067818-A1 CHIMERIC COMPOUND USED FOR TARGETED DEGRADATION OF BCL-2 PROTEIN, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATION THEREOF 江苏恒瑞医药股份有限公司 2024-04-04 WO disclosed