SCHEMBL30857697

SCHEMBL30857697

CC(C)(C)[Si](C)(C)OC[C@]1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN(c3ccc(C(=O)O)cc3)CC2)C1

nearest known ligand 0.69

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BCL2L1 Q07817 12/20 0.69
BCL2 P10415 15/20 0.54
BID P55957 3/20 0.41
BCL2A1 Q16548 3/20 0.41
BCL2L11 O43521 1/20 0.40
CYP2C9 P11712 1/20 0.40
MCL1 Q07820 1/20 0.40
ASPH Q12797 1/20 0.40
BCL2L2 Q92843 1/20 0.40
BAD Q92934 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22325101 0.91 BCL2L1 (0.56) BCL2L1BCL2
SCHEMBL30857610 0.91 BCL2L1 (0.56) BCL2L1BCL2
SCHEMBL25712911 0.85 BCL2L1 (0.81) BCL2L1BCL2BIDBCL2A1
SCHEMBL31759015 0.84 BCL2L1 (0.48) BCL2L1BCL2
SCHEMBL25423208 0.83 BCL2L1 (0.67) BCL2L1BCL2BIDBCL2A1
SCHEMBL25422237 0.83 BCL2L1 (0.67) BCL2L1BCL2BIDBCL2A1
SCHEMBL25274600 0.82 BCL2L1 (0.77) BCL2L1BCL2BIDBCL2A1
SCHEMBL1567421 0.82 BCL2L1 (1.00) BCL2L1BCL2BIDBCL2A1BAD
SCHEMBL25421347 0.82 BCL2L1 (0.68) BCL2L1BCL2BIDBCL2A1
SCHEMBL25422164 0.82 BCL2L1 (0.65) BCL2L1BCL2BIDBCL2A1BCL2L11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024067818-A1 CHIMERIC COMPOUND USED FOR TARGETED DEGRADATION OF BCL-2 PROTEIN, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATION THEREOF 江苏恒瑞医药股份有限公司 2024-04-04 WO disclosed