SCHEMBL30858355

SCHEMBL30858355

C[Si](C)(C)C#CC1=CCN(C(=O)N2CCOCC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.40
GRM5 P41594 2/20 0.39
MEN1 O00255 1/20 0.39
TP53 P04637 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KIT P10721 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2290995 0.83 GRM5 (0.44) GRM5MEN1KMT2AALDH1A1TSHR
SCHEMBL31558715 0.81 GRM5 (0.43) GRM5CYP2C9TSHR
SCHEMBL31558721 0.81 NAMPT (0.44) GRM5MAPT
SCHEMBL31558713 0.80 AKR1C3 (0.50) AKR1C3MEN1TP53KMT2ALMNA
SCHEMBL31558719 0.80 AKR1C3 (0.50) AKR1C3MEN1TP53KMT2ALMNA
SCHEMBL31558707 0.80 GRM5 (0.42) GRM5
SCHEMBL31558712 0.78 GRM5 (0.40) GRM5MEN1KMT2A
SCHEMBL31558699 0.76 NAMPT (0.39) GRM5
SCHEMBL31558705 0.76 NAMPT (0.39) GRM5
SCHEMBL31558697 0.75 GRM5 (0.39) GRM5MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119816496-A Aromatic acetylene derivative and preparation method and application thereof 浙江海正药业股份有限公司 2025-04-11 CN disclosed
WO-2024067812-A1 AROMATIC ACETYLENE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江海正药业股份有限公司 2024-04-04 WO disclosed