Enalapril

Enalapril

SCHEMBL308603

CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1CCC[C@H]1C(=O)O.CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1CCC[C@H]1C(=O)O.O=C(O)/C=C\C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACE

The experimentally established mechanism targets of Enalapril. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACE known ✓ P12821 14/20 0.91
SMN1; SMN2 Q16637 1/20 1.00
LMNA P02545 2/20 0.91
ABCB11 O95342 2/20 0.65
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
USP2 O75604 1/20 0.63
CYP3A4 P08684 1/20 0.63
ALOX15 P16050 1/20 0.63
PDE3A Q14432 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Enalapril SCHEMBL20817249 1.00 SMN1; SMN2 (1.00) SMN1; SMN2ACELMNAABCB11MEN1
Enalapril SCHEMBL10 1.00 SMN1; SMN2 (1.00) SMN1; SMN2ACELMNAABCB11MEN1
Enalapril SCHEMBL2719411 1.00 SMN1; SMN2 (1.00) SMN1; SMN2ACELMNAABCB11MEN1
Enalapril SCHEMBL9 1.00 SMN1; SMN2 (1.00) SMN1; SMN2ACELMNAABCB11MEN1
Enalapril SCHEMBL6155137 1.00 SMN1; SMN2 (1.00) SMN1; SMN2ACELMNAABCB11MEN1
Enalapril SCHEMBL10390115 1.00 SMN1; SMN2 (1.00) SMN1; SMN2ACELMNAABCB11MEN1
Enalapril SCHEMBL1650291 1.00 SMN1; SMN2 (1.00) SMN1; SMN2ACELMNAABCB11MEN1
Enalapril SCHEMBL825430 1.00 SMN1; SMN2 (1.00) SMN1; SMN2ACELMNAABCB11MEN1
Enalapril SCHEMBL9019924 0.99 SMN1; SMN2 (0.98) SMN1; SMN2ACELMNAABCB11MEN1
Enalapril SCHEMBL9019927 0.99 SMN1; SMN2 (0.98) SMN1; SMN2ACELMNAABCB11MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3380522-A1 ANTIBODY MOLECULES TO APRIL AND USES THEREOF Visterra, Inc. (US) 2018-10-03 EP disclosed
WO-2017091683-A1 ANTIBODY MOLECULES TO APRIL AND USES THEREOF Visterra, Inc. (US) 2017-06-01 WO disclosed
US-20150366813-A1 LIQUID-FILLED IMMEDIATE RELEASE SOFT GELATIN CAPSULES PATHEON SOFTGELS INC 2015-12-24 US disclosed
WO-2015195990-A1 LIQUID-FILLED IMMEDIATE RELEASE SOFT GELATIN CAPSULES BANNER LIFE SCIENCES LLC (US) 2015-12-23 WO disclosed
EP-2736489-A1 COMPOSITIONS, PROCESS OF PREPARATION OF SAID COMPOSITIONS AND METHOD OF TREATING INFLAMMATORY DISEASES Cellworks Research India Private Limited (IN) 2014-06-04 EP disclosed
WO-2013016718-A1 COMPOSITIONS, PROCESS OF PREPARATION OF SAID COMPOSITIONS AND METHOD OF TREATING INFLAMMATORY DISEASES CELLWORKS RESEARCH INDIA PRIVATE LIMITED (IN) 2013-01-31 WO disclosed
US-20120101630-A1 PHARMACEUTICAL PACKAGING AND METHOD FOR DELIVERY OF SAME DAYA MEDICALS, INC. 2012-04-26 US disclosed
EP-2434017-A2 Identification of a micro-RNA that activates expression of beta-myosin heavy chain Board of Regents of the University of Texas System (US) 2012-03-28 EP disclosed
US-20120040902-A1 METHOD OF TREATING DYSPNEA ASSOCIATED WITH ACUTE HEART FAILURE UNEMORI ELAINE (US) 2012-02-16 US disclosed
US-20120040903-A1 METHOD FOR TREATING DYSPNEA ASSOCIATED WITH ACUTE HEART FAILURE CORTHERA, INC. 2012-02-16 US disclosed
WO-2011044377-A2 CHELATOR-TARGETING LIGAND CONJUGATES FOR CARDIOVASCULAR IMAGING CELL POINT, LLC (US) 2011-04-14 WO disclosed
US-20110085969-A1 CHELATOR-TARGETING LIGAND CONJUGATES FOR CARDIOVASCULAR IMAGING CELL>POINT, LLC 2011-04-14 US disclosed
EP-2102214-B1 4, 5, 6, 7-TETRAHYDRO-THIENO [3, 2-C] PYRIDINE DERIVATIVES AS H3 MODULATORS HOFFMANN LA ROCHE (CH) 2011-03-23 EP disclosed
US-7902184-B2 Piperazinyl pyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-03-08 US disclosed
EP-2288366-A2 METHOD OF TREATING CHRONIC HEART FAILURE Corthera, Inc. (US) 2011-03-02 EP disclosed
EP-2288373-A2 TREATING DYSPNEA ASSOCIATED WITH ACUTE HEART FAILURE WITH RELAXIN Corthera, Inc. (US) 2011-03-02 EP disclosed
EP-1957479-B1 1,5-SUBSTITUTED INDOL-2-YL AMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-03-02 EP disclosed
WO-2011011114-A2 PHARMACEUTICAL PACKAGING AND METHOD FOR DELIVERY OF SAME DAYA MEDICALS, INC. (US) 2011-01-27 WO disclosed
WO-2002087503-A2 COMPOSITIONS AND METHODS FOR TREATING COLORECTAL POLYPS AND CANCER VANDERBILT UNIVERSITY (US) 2002-11-07 WO disclosed
WO-2002059343-A2 BIOLOGICAL MARKERS AND DIAGNOSTIC TESTS FOR ANGIOTENSIN CONVERTING ENZYME INHIBITOR- AND VASOPEPTIDASE INHIBITOR-ASSOCIATED ANGIOEDEMA VANDERBILT UNIVERSITY (US) 2002-08-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110085969-A1 CHELATOR-TARGETING LIGAND CONJUGATES FOR CARDIOVASCULAR IMAGING SLC2A8, SLC2A1, SLC2A2 ACE 1634/4885SMN1; SMN2 2522/4885LMNA 4179/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.