SCHEMBL30870569

SCHEMBL30870569

Cc1ccc(N=C=O)cc1C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.58
TRPA1 O75762 1/20 0.58
MAPK1 P28482 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TSHR P16473 1/20 0.37
NOTUM Q6P988 1/20 0.37
TAS2R14 Q9NYV8 1/20 0.35
ALKBH5 Q6P6C2 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
S1PR1 P21453 4/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
CYP1A2 P05177 1/20 0.32
USP30 Q70CQ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1403637 1.00 CYP3A4 (0.58) CYP3A4TRPA1MAPK1TDP1TSHR
SCHEMBL22815461 0.84 CYP3A4 (0.59) CYP3A4TRPA1MAPK1TDP1TSHR
SCHEMBL1555041 0.83 MAPK1 (0.47) CYP3A4TRPA1MAPK1TDP1TSHR
SCHEMBL13813270 0.82 P2RY6 (0.37) CYP3A4TRPA1TDP1NOTUMTAS2R14
SCHEMBL29069269 0.82 CYP3A4 (0.58) CYP3A4TRPA1MAPK1TDP1TSHR
SCHEMBL7177146 0.81 MAPK1 (0.46) CYP3A4TRPA1MAPK1TDP1TSHR
SCHEMBL3104369 0.80 CYP3A4 (0.50) CYP3A4TRPA1MAPK1TDP1TSHR
SCHEMBL29648906 0.80 MAPK1 (0.44) CYP3A4TRPA1MAPK1TDP1TSHR
SCHEMBL60206 0.80 MAPK1 (0.44) CYP3A4TRPA1MAPK1TDP1TSHR
SCHEMBL12367734 0.79 NOTUM (0.40) CYP3A4TRPA1MAPK1TSHRNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112074511-B Substituted benzodiazoles and their use in therapy 托马斯·黑勒戴药物研究基金会 2024-04-26 CN disclosed