SCHEMBL30872018

SCHEMBL30872018

CC(=O)n1ccc2cccc(N)c21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.53
ALDH1A1 P00352 4/20 0.40
HPGD P15428 4/20 0.40
KDM4E B2RXH2 3/20 0.40
HSD17B10 Q99714 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
PARP1 P09874 1/20 0.37
CYP11B1 P15538 3/20 0.35
CYP11B2 P19099 3/20 0.35
TSHR P16473 4/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
OXER1 Q8TDS5 1/20 0.35
TP53 P04637 1/20 0.33
GLA P06280 1/20 0.33
CYP3A4 P08684 2/20 0.32
KEAP1 Q14145 1/20 0.32
HRH4 Q9H3N8 1/20 0.32
MMP2 P08253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29216392 1.00 NOTUM (0.53) NOTUMALDH1A1HPGDKDM4EHSD17B10
SCHEMBL21055089 0.84 TSHR (0.40) NOTUMALDH1A1HPGDHSD17B10KMT2A
SCHEMBL29216394 0.81 OXER1 (0.43) NOTUMALDH1A1KDM4EHSD17B10MEN1
SCHEMBL30872017 0.81 OXER1 (0.43) NOTUMALDH1A1KDM4EHSD17B10MEN1
SCHEMBL10836512 0.79 NOTUM (0.56) NOTUMALDH1A1HPGDKDM4EHSD17B10
SCHEMBL21055656 0.78 ACLY (0.47) NOTUML3MBTL1PIK3CA
SCHEMBL30826403 0.76 NOTUM (0.50) NOTUMALDH1A1HPGDKDM4EHSD17B10
SCHEMBL29187805 0.76 NOTUM (0.50) NOTUMALDH1A1HPGDKDM4EHSD17B10
SCHEMBL13139572 0.75 KMT2A (0.39) NOTUMALDH1A1HPGDKDM4EHSD17B10
SCHEMBL30847966 0.71 PRKCI (0.39) ALDH1A1HPGDHSD17B10TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117794914-A Pyrimidine-2, 4-diamine derivatives, process for preparing the same, and pharmaceutical composition for preventing or treating cancer comprising the same as active ingredient 韩国化学研究院 2024-03-29 CN disclosed