SCHEMBL30872091

SCHEMBL30872091

N#Cc1ccc(-c2ccncn2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.54
CYP2D6 P10635 1/20 0.51
CYP11B2 P19099 1/20 0.46
CYP11B1 P15538 1/20 0.44
KDM1A O60341 1/20 0.43
GAA P10253 1/20 0.42
EGLN2 Q96KS0 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
HTT P42858 1/20 0.41
CDC7 O00311 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MMP3 P08254 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24791664 1.00 GRM5 (0.54) GRM5CYP2D6CYP11B2CYP11B1KDM1A
SCHEMBL9903935 0.83 CYP2D6 (0.60) GRM5CYP2D6GSK3AGSK3BMAP4K4
SCHEMBL18889616 0.79 GRM5 (0.83) GRM5CYP2D6CYP11B1KDM1AEGLN2
SCHEMBL6847956 0.78 CYP2D6 (0.49) GRM5CYP2D6GSK3AGSK3BMAP4K4
SCHEMBL13986853 0.78 KDM4E (0.59) GRM5CYP11B2CYP11B1KDM1AGAA
SCHEMBL31108745 0.77 GRM5 (0.51) GRM5CYP11B2CYP11B1KDM1AEGLN2
SCHEMBL5145719 0.77 GRM5 (0.51) GRM5CYP11B2CYP11B1KDM1AEGLN2
SCHEMBL8499115 0.77 CYP2D6 (0.53) GRM5CYP2D6GSK3B
SCHEMBL28801114 0.77 GRM5 (0.54) GRM5CYP2D6CYP11B2CYP11B1EGLN2
SCHEMBL29394412 0.76 GRM5 (0.84) GRM5CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117940427-A Substituted pyrazolo [1,5-a ] pyrimidine-7-amine compounds as CDK inhibitors and therapeutic uses thereof 卡里克治疗有限公司 2024-04-26 CN disclosed