SCHEMBL30872207

SCHEMBL30872207

CCS(=O)(=O)OO[C@H]1CN(C(c2ccccc2)c2ccccc2)[C@@H]1C

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 4/20 0.41
SLC6A9 P48067 1/20 0.39
SIGMAR1 Q99720 2/20 0.36
KDM4E B2RXH2 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
HPGD P15428 2/20 0.36
CYP2C19 P33261 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5458868 0.82 OPRD1 (0.38) OPRD1SLC6A9CYP3A4CYP2C9CYP2C19
SCHEMBL30642715 0.82 OPRD1 (0.38) OPRD1SLC6A9CYP3A4CYP2C9CYP2C19
SCHEMBL5450723 0.82 OPRD1 (0.38) OPRD1SLC6A9CYP3A4CYP2C9CYP2C19
SCHEMBL5458873 0.82 OPRD1 (0.38) OPRD1SLC6A9CYP3A4CYP2C9CYP2C19
SCHEMBL30733235 0.77 OPRD1 (0.42) OPRD1SLC6A9KDM4ECYP1A2CYP3A4
SCHEMBL2769798 0.76 OPRD1 (0.42) OPRD1SIGMAR1
SCHEMBL14671934 0.76 OPRD1 (0.42) OPRD1SIGMAR1
SCHEMBL14663826 0.76 OPRD1 (0.42) OPRD1SIGMAR1
SCHEMBL14663829 0.76 OPRD1 (0.42) OPRD1SIGMAR1
SCHEMBL14663828 0.76 OPRD1 (0.42) OPRD1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117881670-A Methods of making EGFR inhibitors 缆图药品公司 2024-04-12 CN disclosed