SCHEMBL30873286

SCHEMBL30873286

CSc1nc(NC(C)(C)C)ncc1Br

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 8/20 0.38
CDK2 P24941 8/20 0.38
KDR P35968 5/20 0.38
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
CCND2 P30279 1/20 0.35
CCND3 P30281 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
ALDH1A1 P00352 1/20 0.32
RAB9A P51151 1/20 0.32
GAA P10253 1/20 0.31
LRRK2 Q5S007 1/20 0.30
CYP1A2 P05177 1/20 0.30
PDE4A P27815 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13734929 1.00 CDK1 (0.38) CDK1CDK2KDRCDK4CCND1
SCHEMBL23196010 0.81 CDK4 (0.36) KDRCDK4CCND1CCND2CCND3
SCHEMBL23195815 0.79 SMN1; SMN2 (0.41) CDK2CDK4CCND1CCND2CCND3
SCHEMBL23195809 0.76 IGF1R (0.40) CDK1CDK2KDRCDK4CCND1
SCHEMBL13733999 0.76 KDM4E (0.37) CDK1KDRCDK4CCND1CCND2
SCHEMBL23196386 0.74 MAPK8 (0.39) CDK4CCND1CCND2CCND3SMN1; SMN2
SCHEMBL13734259 0.73 MAPK8 (0.48)
SCHEMBL13734497 0.72 HDAC3 (0.38) CDK1CDK2KDRLRRK2
SCHEMBL4584347 0.70 IGF1R (0.48) CDK1CDK2KDR
SCHEMBL3450501 0.70 HDAC3 (0.44) CDK1CDK2KDRCDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111471021-B Substituted diamino carboxamides and diamino carbonitrile pyrimidines, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2024-04-02 CN disclosed