SCHEMBL30874372

SCHEMBL30874372

Cc1ccc([N+](=O)[O-])c2c(=O)n(CC(=O)O)ccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B10 O60218 1/20 0.40
AKR1B1 P15121 1/20 0.40
RAD52 P43351 1/20 0.38
TSHR P16473 2/20 0.38
POLB P06746 3/20 0.36
KMT2A Q03164 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MEN1 O00255 1/20 0.36
CASP6 P55212 1/20 0.36
TLR9 Q9NR96 1/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
GAA P10253 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
ELANE P08246 1/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7234130 0.72 RAD52 (0.56) AKR1B10AKR1B1RAD52TSHRKMT2A
SCHEMBL3165711 0.69 KMT2A (0.50) AKR1B10AKR1B1KMT2AALDH1A1KDM4E
SCHEMBL21685452 0.68 TSHR (0.41) AKR1B10AKR1B1TSHRKMT2AL3MBTL1
SCHEMBL21685619 0.67 ALDH1A1 (0.47) AKR1B10AKR1B1TSHRPOLBALDH1A1
SCHEMBL7604837 0.67 TSHR (0.43) TSHRPOLBKMT2AL3MBTL1MEN1
SCHEMBL4592116 0.65 MAPT (0.49) POLBKMT2AMEN1ALDH1A1KDM4E
SCHEMBL12875609 0.64 KMT2A (0.56) KMT2AMEN1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL27757531 0.63 ALDH1A1 (0.48) POLBKMT2AMEN1ALDH1A1KDM4E
SCHEMBL1590530 0.63 GAA (0.56) RAD52TSHRKMT2AMEN1ALDH1A1
SCHEMBL2875153 0.63 KMT2A (0.50) AKR1B10AKR1B1TSHRKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117813297-A Phenyl and pyridopyrazole derivatives as DDR1 inhibitors 莱德克斯制药公共有限公司 2024-04-02 CN disclosed