SCHEMBL30878308

SCHEMBL30878308

C#Cc1cc(=O)n(-c2ccc(NC(=O)CC)cc2)c2nc(Nc3ccccc3OC)ncc12

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 3/20 0.52
BTK Q06187 2/20 0.47
EGFR P00533 12/20 0.46
JAK3 P52333 3/20 0.46
AKT3 Q9Y243 1/20 0.44
MAP4K1 Q92918 1/20 0.44
TTK P33981 3/20 0.43
BLK P51451 2/20 0.43
NUAK1 O60285 1/20 0.43
NUAK2 Q9H093 1/20 0.43
GAK O14976 1/20 0.43
ERBB2 P04626 1/20 0.43
JAK1 P23458 1/20 0.43
TXK P42681 1/20 0.43
ITK Q08881 1/20 0.43
ERBB4 Q15303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30878486 0.92 FLT3 (0.51) FLT3BTKEGFRJAK3MAP4K1
SCHEMBL30879348 0.92 MAPK3 (0.49) FLT3BTKEGFRJAK3MAP4K1
SCHEMBL30878477 0.91 EGFR (0.51) FLT3BTKEGFRJAK3AKT3
SCHEMBL30878392 0.89 BTK (0.61) FLT3BTKEGFRJAK3BLK
SCHEMBL30878733 0.88 FLT3 (0.48) FLT3BTKEGFRJAK3AKT3
SCHEMBL30878716 0.88 FLT3 (0.48) FLT3BTKEGFRJAK3AKT3
SCHEMBL30878470 0.87 MAP4K1 (0.55) BTKEGFRJAK3MAP4K1
SCHEMBL30878437 0.86 MAP4K1 (0.54) FLT3BTKEGFRMAP4K1BLK
SCHEMBL30878482 0.86 MAP4K1 (0.52) FLT3BTKEGFRMAP4K1BLK
SCHEMBL30878336 0.85 FLT3 (0.51) FLT3BTKEGFRMAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP claimed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO claimed
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP disclosed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO disclosed