SCHEMBL30878690

SCHEMBL30878690

COc1ccccc1-c1c(C#C[Si](C(C)C)(C(C)C)C(C)C)c2cnc(Nc3ccc(N(C)CCN(C)C)cc3)nc2n(C)c1=O

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 1/20 0.43
EGFR P00533 7/20 0.41
BTK Q06187 2/20 0.41
WEE1 P30291 7/20 0.41
CCNT1 O60563 2/20 0.41
CDK9 P50750 2/20 0.41
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
FGFR1 P11362 4/20 0.40
SRC P12931 2/20 0.38
JAK3 P52333 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30879233 0.90 WEE1 (0.52) FGFR4EGFRWEE1CCNT1CDK9
SCHEMBL30878353 0.89 FGFR4 (0.47) FGFR4EGFRBTKWEE1CCNT1
SCHEMBL30879105 0.86 FGFR1 (0.46) FGFR4EGFRBTKWEE1CCNT1
SCHEMBL30879282 0.86 FGFR1 (0.42) FGFR4EGFRWEE1CCNT1CDK9
SCHEMBL30879066 0.85 FGFR1 (0.48) FGFR4EGFRBTKWEE1CCNT1
SCHEMBL30879162 0.85 EGFR (0.48) FGFR4EGFRBTKWEE1CDK4
SCHEMBL30879118 0.85 WEE1 (0.42) FGFR4EGFRBTKWEE1CCNT1
SCHEMBL30878874 0.84 FGFR1 (0.43) FGFR4EGFRBTKWEE1CCNT1
SCHEMBL30879314 0.84 CCNT1 (0.44) FGFR4EGFRBTKWEE1CCNT1
SCHEMBL30878727 0.83 EGFR (0.50) FGFR4EGFRBTKCDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4612148-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER Cancer Research Technology Limited (GB) 2025-09-10 EP disclosed
WO-2024094963-A1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE AND 7-AMINO-1-PYRIMIDO[4,5-D]PYRIMIDIN-2(1 H)-ONE DERIVATIVES AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2024-05-10 WO disclosed