SCHEMBL30880666

SCHEMBL30880666

COc1cc(Nc2ccnc3ccccc23)cc(-n2ccnc2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.60
GAK O14976 6/20 0.55
RIPK2 O43353 3/20 0.55
COQ8A Q8NI60 3/20 0.55
NLK Q9UBE8 3/20 0.55
ERBB2 P04626 1/20 0.49
ADRA2A P08913 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
MITF O75030 1/20 0.44
RAD52 P43351 1/20 0.44
FADS1 O60427 1/20 0.44
EGFR P00533 1/20 0.44
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
MAPKAPK2 P49137 1/20 0.42
LMNA P02545 1/20 0.41
HDAC3 O15379 1/20 0.41
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30880707 0.89 GAK (0.58) HTTGAKRIPK2COQ8ANLK
SCHEMBL30880458 0.89 GAK (0.58) HTTGAKRIPK2COQ8ANLK
SCHEMBL30880722 0.88 RIPK2 (0.49) HTTGAKRIPK2COQ8ANLK
SCHEMBL30880531 0.87 GAK (0.58) HTTGAKRIPK2COQ8ANLK
SCHEMBL30880617 0.87 GAK (0.58) HTTGAKRIPK2COQ8ANLK
SCHEMBL30880628 0.86 GAK (0.57) HTTGAKRIPK2COQ8ANLK
SCHEMBL30880499 0.86 GAK (0.57) HTTGAKRIPK2COQ8ANLK
SCHEMBL30880737 0.86 GAK (0.57) HTTGAKRIPK2COQ8ANLK
SCHEMBL30880564 0.86 GAK (0.57) HTTGAKRIPK2COQ8ANLK
SCHEMBL30880581 0.86 GAK (0.57) GAKRIPK2COQ8ANLKADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024078513-A1 CONDENSED AZINES FOR TREATING CANCER CHENGDU ANTICANCER BIOSCIENCE , LTD. (CN) 2024-04-18 WO disclosed