Ajmaline

Ajmaline

SCHEMBL30892623

CC[C@H]1[C@@H]2C[C@H]3[C@@H]4N(C)c5ccccc5[C@]45C[C@@H]([C@H]2[C@H]5O)N3[C@@H]1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 1.00
KCNH2 Q12809 2/20 1.00
SCN5A Q14524 2/20 1.00
KMT2A Q03164 2/20 1.00
ADRA2B P18089 1/20 1.00
ADRA2C P18825 1/20 1.00
DRD3 P35462 1/20 1.00
OPRK1 P41145 1/20 1.00
MEN1 O00255 1/20 1.00
TSHR P16473 1/20 1.00
CACNA1F O60840 1/20 1.00
SCN1A P35498 1/20 1.00
SCN4A P35499 1/20 1.00
SCN7A Q01118 1/20 1.00
CACNA1D Q01668 1/20 1.00
CACNA1S Q13698 1/20 1.00
CACNA1C Q13936 1/20 1.00
SCN9A Q15858 1/20 1.00
SCN2A Q99250 1/20 1.00
SCN3A Q9NY46 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ajmaline SCHEMBL29620363 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B
Ajmaline SCHEMBL30116336 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B
Ajmaline SCHEMBL29811209 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B
Ajmaline SCHEMBL14029381 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B
Ajmaline SCHEMBL2787287 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B
Ajmaline SCHEMBL23295973 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B
Ajmaline SCHEMBL10422895 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B
Ajmaline SCHEMBL29354066 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B
Ajmaline SCHEMBL15384531 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B
Ajmaline SCHEMBL18950 1.00 CYP2D6 (1.00) CYP2D6KCNH2SCN5AKMT2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111246873-B Optimized peptides for targeting human nerves and their use in image guided surgery, diagnosis and therapy delivery 加利福尼亚大学董事会 2024-03-01 CN disclosed