SCHEMBL30895267

SCHEMBL30895267

Cc1nn(C(F)(F)F)c2ccc(Br)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.39
ADORA2A P29274 2/20 0.35
ADORA2B P29275 2/20 0.35
NT5E P21589 1/20 0.34
CASP3 P42574 2/20 0.34
PDE2A O00408 1/20 0.33
ELANE P08246 3/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
IDO1 P14902 1/20 0.32
LMNA P02545 2/20 0.32
TP53 P04637 1/20 0.32
HAVCR2 Q8TDQ0 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
PDGFRA P16234 1/20 0.32
CDK5 Q00535 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30895272 0.87 PDGFRA (0.38) MAPK8ADORA2AADORA2BNT5ECASP3
SCHEMBL30895271 0.87 PDGFRA (0.38) MAPK8ADORA2AADORA2BNT5ECASP3
SCHEMBL17177295 0.85 MAPK8 (0.40) MAPK8ADORA2AADORA2BCASP3ELANE
SCHEMBL28245972 0.77 NT5E (0.41) NT5ECASP3LMNACYP1A2CYP2D6
SCHEMBL1336984 0.75 ADORA2A (0.59) MAPK8ADORA2AADORA2BCASP3NPC1
SCHEMBL23535755 0.73 MAPK8 (0.39) MAPK8ADORA2AADORA2BCASP3ELANE
SCHEMBL15970798 0.71 MAPK8 (0.40) MAPK8ADORA2AADORA2BCASP3ELANE
SCHEMBL30895247 0.71 IDO1 (0.38) IDO1
SCHEMBL20176288 0.70 MAPK8 (0.39) MAPK8ADORA2AADORA2BCASP3ELANE
SCHEMBL5316056 0.70 MAPK8 (0.39) MAPK8ADORA2AADORA2BCASP3ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4608507-A1 COMPOUNDS AND COMPOSITIONS AS GPR52 MODULATORS Neurocrine Biosciences, Inc. (US) 2025-09-03 EP disclosed
WO-2024091538-A1 COMPOUNDS AND COMPOSITIONS AS GPR52 MODULATORS NEUROCRINE BIOSCIENCES, INC. (US) 2024-05-02 WO disclosed