SCHEMBL30900413

SCHEMBL30900413

CC(C)(C)OC(=O)N1C(=O)c2cc(Br)sc2C12CC2

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.33
BUB1 O43683 1/20 0.33
FPR3 P25089 1/20 0.31
FPR2 P25090 1/20 0.31
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
GSK3B P49841 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31
GPR119 Q8TDV5 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
PIK3R1 P27986 1/20 0.30
PIK3CA P42336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17837270 0.85 BUB1 (0.34) ELANEBUB1CCNB2CDK1CCNB1
SCHEMBL30900353 0.78 BUB1 (0.37) ELANEBUB1FPR3FPR2GPR119
SCHEMBL30900382 0.72 CCND1 (0.32)
SCHEMBL25349215 0.72
SCHEMBL1806153 0.70 AVPR1A (0.40) GPR119KDM4EMAPTTHRB
SCHEMBL21075868 0.69 BUB1 (0.34) ELANEBUB1
SCHEMBL22470779 0.69
SCHEMBL25349493 0.67 BACE1 (0.32)
SCHEMBL31411821 0.67 BCHE (0.39) BUB1CDK1
SCHEMBL23481064 0.66 USP2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117658987-A Compounds as PLK1 inhibitors, and preparation method and application thereof 上海深势唯思科技有限责任公司 2024-03-08 CN disclosed