SCHEMBL30916111

SCHEMBL30916111

O=Cc1nc2c(s1)CN(C1COC1)CC2

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.40
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
PDE1B Q01064 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23109923 0.75 RAD52 (0.40) GRM5PDCD1CD274PDE1BKCNH2
SCHEMBL14925519 0.75 GRM5 (0.40) GRM5PDCD1CD274PDE1BKCNH2
Lithium Ion SCHEMBL27175184 0.75 GRM5 (0.38) GRM5PDCD1CD274PDE1BKCNH2
SCHEMBL24538478 0.70 PDCD1 (0.36) GRM5PDCD1CD274
SCHEMBL30916103 0.68 RAD52 (0.41) GRM5
SCHEMBL23699915 0.67 PDK1 (0.56)
SCHEMBL30916117 0.67 RAD52 (0.40) GRM5
SCHEMBL14817814 0.65 GRM5 (0.32) GRM5
SCHEMBL24585187 0.65 CYP3A4 (0.45)
SCHEMBL18375024 0.65 GRM5 (0.38) GRM5PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111936475-B Immunomodulator, composition and preparation method thereof 贝达药业股份有限公司 2024-05-10 CN claimed
CN-111936475-B Immunomodulator, composition and preparation method thereof 贝达药业股份有限公司 2024-05-10 CN disclosed