SCHEMBL30919449

SCHEMBL30919449

Cc1nn(-c2ccc(NC(=O)OC(C)(C)C)cn2)cc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
BCL2 P10415 2/20 0.40
HDAC3 O15379 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
MAPKAPK2 P49137 3/20 0.38
CYP17A1 P05093 2/20 0.37
BRD4 O60885 1/20 0.37
MAPK14 Q16539 1/20 0.36
RORC P51449 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA9 Q16790 1/20 0.36
PSMB8 P28062 1/20 0.36
MAP4K4 O95819 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
BECN1 Q14457 1/20 0.35
WNT3A P56704 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24896788 1.00 NAMPT (0.41) NAMPTPTGDR2BCL2HDAC3HDAC8
SCHEMBL25255538 0.87 NAMPT (0.39) NAMPTPTGDR2BCL2HDAC3HDAC8
SCHEMBL25253508 0.86 MAPKAPK2 (0.41) NAMPTPTGDR2BCL2HDAC3HDAC8
SCHEMBL25255285 0.85 AR (0.41) NAMPTPTGDR2BCL2HDAC3HDAC8
SCHEMBL25413782 0.84 MAPT (0.38) KDM4EMAPT
SCHEMBL26453252 0.79 PTGDR2 (0.36) NAMPTPTGDR2MAPKAPK2BRD4RORC
SCHEMBL30362248 0.79 PTGDR2 (0.38) NAMPTPTGDR2HDAC3HDAC8NCOR2
SCHEMBL25251320 0.79 PTGDR2 (0.38) NAMPTPTGDR2HDAC3HDAC8NCOR2
SCHEMBL24896789 0.79 PTGDR2 (0.36) NAMPTPTGDR2MAPKAPK2CYP17A1BRD4
SCHEMBL30919455 0.79 PTGDR2 (0.36) NAMPTPTGDR2MAPKAPK2CYP17A1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118119609-A Imidazole derivatives and their use as antibiotics 豪夫迈·罗氏有限公司 2024-05-31 CN disclosed