Bromide

Bromide

SCHEMBL30920113

Br.CCOC(=O)C1NCCc2cc(O)ccc21

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
ESR1 P03372 2/20 0.41
ESR2 Q92731 2/20 0.41
KMT2A Q03164 1/20 0.40
HSD17B1 P14061 2/20 0.39
BCHE P06276 1/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM1A O60341 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
KIF11 P52732 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL28658741 1.00 CA1 (0.43) CA1CA2CA7CA9CA14
SCHEMBL8259309 0.99 CA1 (0.43) CA1CA2CA7CA9CA14
Hydrochloric Acid SCHEMBL8298614 0.97 CA1 (0.43) CA1CA2CA7CA9CA14
SCHEMBL4478957 0.90 NQO2 (0.41) CA1CA2CA7CA9CA14
SCHEMBL19960840 0.85 ALDH1A1 (0.40) CA1CA2CA7CA9CA14
SCHEMBL7124159 0.84 CA1 (0.46) CA1CA2CA7CA9CA14
SCHEMBL10516146 0.84 KMT2A (0.48) CA1CA2CA7CA9CA14
Hydrochloric Acid SCHEMBL19953589 0.84 TSHR (0.41) CA1CA2CA7CA9CA14
Hydrochloric Acid SCHEMBL3534709 0.83 CA1 (0.45) CA1CA2CA7CA9CA14
SCHEMBL23119015 0.81 TSHR (0.60) TSHRNPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118580188-A Can be used as ROR gamma regulator aniline compound (B) 励缔(杭州)医药科技有限公司 2024-09-03 CN disclosed
CN-113773251-B Anilines useful as rory modulators 励缔(杭州)医药科技有限公司 2024-06-11 CN disclosed
CN-113666863-B Biaryl compounds useful as rory modulators 励缔(杭州)医药科技有限公司 2024-06-11 CN disclosed