SCHEMBL30926482

SCHEMBL30926482

CC(C)(C)c1cnc2ccc(Br)cn12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.43
MTOR P42345 1/20 0.43
MAP3K14 Q99558 1/20 0.43
GAA P10253 1/20 0.43
SCN5A Q14524 1/20 0.37
FLT3 P36888 2/20 0.36
TSHR P16473 1/20 0.36
MAPK10 P53779 1/20 0.36
ADORA2A P29274 1/20 0.34
TRIM33 Q9UPN9 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
PIK3CD O00329 1/20 0.33
DYRK3 O43781 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK2 P24941 1/20 0.33
CSNK1E P49674 1/20 0.33
CLK1 P49759 1/20 0.33
CLK2 P49760 1/20 0.33
CLK3 P49761 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15639933 0.82 SCN5A (0.54) PIK3CAMTORMAP3K14GAASCN5A
SCHEMBL24654977 0.80 CYP1A2 (0.50) MAP3K14GAASCN5A
SCHEMBL23419244 0.80 SCN5A (0.38) SCN5ATSHRMAP3K5EIF2AK4
SCHEMBL21305144 0.79 POLB (0.51) MAP3K14GAASCN5AFLT3PIK3CD
SCHEMBL12998303 0.76 PIK3CA (0.47) PIK3CAMTORMAP3K14GAAFLT3
SCHEMBL3029604 0.75 MAP3K14 (0.49) PIK3CAMTORMAP3K14GAAFLT3
SCHEMBL30926487 0.75 SCN5A (0.35) SCN5A
SCHEMBL16011333 0.75 GAA (0.54) PIK3CAMTORMAP3K14GAAFLT3
SCHEMBL21370423 0.73 SCN5A (0.35) SCN5AEIF2AK4
SCHEMBL19631457 0.73 CYP1A2 (0.42) GAASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4626423-A1 CDK INHIBITORS AND METHODS AND USE THEREOF Relay Therapeutics, Inc. (US) 2025-10-08 EP disclosed
WO-2024119122-A1 CDK INHIBITORS AND METHODS AND USE THEREOF RELAY THERAPEUTICS, INC. (US) 2024-06-06 WO disclosed