SCHEMBL30928261

SCHEMBL30928261

COc1cc(/C=C/C(=O)/C=C/c2cc(Br)c(O)c(OC)c2)cc(Br)c1O

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.80
KDM4E B2RXH2 1/20 0.80
CYP1A2 P05177 2/20 0.78
CYP2D6 P10635 2/20 0.78
CYP3A4 P08684 1/20 0.78
CYP2C9 P11712 1/20 0.78
CYP2B6 P20813 1/20 0.78
ALOX5 P09917 6/20 0.68
STAT3 P40763 4/20 0.68
NFKB1 P19838 3/20 0.68
NFKB2 Q00653 3/20 0.68
RELA Q04206 3/20 0.68
NFE2L2 Q16236 3/20 0.68
PTGS1 P23219 2/20 0.61
PTGS2 P35354 2/20 0.61
PKM P14618 1/20 0.61
PTGES O14684 2/20 0.58
HSD11B1 P28845 1/20 0.58
PRMT1 Q99873 1/20 0.56
LY96 Q9Y6Y9 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30928252 1.00 GAA (0.80) GAAKDM4ECYP1A2CYP2D6CYP3A4
SCHEMBL30966316 0.89 KDM4E (1.00) GAAKDM4ECYP1A2CYP2D6CYP3A4
SCHEMBL31207225 0.89 KDM4E (1.00) GAAKDM4ECYP1A2CYP2D6CYP3A4
SCHEMBL29242003 0.89 KDM4E (1.00) GAAKDM4ECYP1A2CYP2D6CYP3A4
SCHEMBL2743839 0.88 CYP1A2 (1.00) GAAKDM4ECYP1A2CYP2D6CYP3A4
SCHEMBL2743841 0.88 CYP1A2 (1.00) GAAKDM4ECYP1A2CYP2D6CYP3A4
SCHEMBL14875151 0.88 KDM4E (0.76) GAAKDM4ECYP1A2CYP2D6CYP3A4
SCHEMBL14875150 0.88 KDM4E (0.76) GAAKDM4ECYP1A2CYP2D6CYP3A4
SCHEMBL16454768 0.82 PRMT1 (0.77) GAAKDM4ECYP1A2CYP2D6CYP3A4
SCHEMBL30179914 0.82 CYP1A2 (0.87) GAAKDM4ECYP1A2CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084645-A Conjugated ketene skeleton bromophenol compound, preparation method and anti-tumor application 中国海洋大学 2024-05-28 CN claimed