SCHEMBL30928263

SCHEMBL30928263

COc1cc(C=CC(=O)C=Cc2cc(OC)c(O)c(Br)c2Br)c(Br)c(Br)c1O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 5/20 0.60
CYP1A2 P05177 2/20 0.58
CYP2D6 P10635 2/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2B6 P20813 1/20 0.58
NFKB1 P19838 4/20 0.51
ALOX5 P09917 3/20 0.51
STAT3 P40763 3/20 0.51
NFKB2 Q00653 3/20 0.51
RELA Q04206 3/20 0.51
LY96 Q9Y6Y9 3/20 0.50
MAPT P10636 2/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
KMT2A Q03164 1/20 0.50
JUN P05412 1/20 0.50
TFEB P19484 1/20 0.50
KDM4E B2RXH2 2/20 0.48
NPC1 O15118 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31366778 0.81 NFE2L2 (0.54) NFE2L2CYP1A2CYP2D6CYP3A4CYP2C9
SCHEMBL30928251 0.81 NFE2L2 (0.54) NFE2L2CYP1A2CYP2D6CYP3A4CYP2C9
SCHEMBL1646879 0.80 ERN1 (0.64) MAPTALDH1A1KDM4ETDP1ERN1
SCHEMBL16093497 0.79 NFE2L2 (0.62) NFE2L2CYP1A2CYP2D6CYP3A4CYP2C9
SCHEMBL16385977 0.79 NFE2L2 (0.62) NFE2L2CYP1A2CYP2D6CYP3A4CYP2C9
SCHEMBL1647147 0.79 BACE1 (0.71) CYP2D6CYP2C9MAPTPTGS2
SCHEMBL1647144 0.79 BACE1 (0.71) CYP2D6CYP2C9MAPTPTGS2
SCHEMBL30928257 0.78 NFE2L2 (0.71) NFE2L2CYP1A2CYP2D6CYP3A4CYP2C9
SCHEMBL30928256 0.77 BACE1 (0.64) NFE2L2CYP1A2CYP2D6CYP3A4CYP2C9
SCHEMBL2744657 0.75 NFE2L2 (1.00) NFE2L2CYP1A2CYP2D6CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084645-A Conjugated ketene skeleton bromophenol compound, preparation method and anti-tumor application 中国海洋大学 2024-05-28 CN claimed
CN-118084645-A Conjugated ketene skeleton bromophenol compound, preparation method and anti-tumor application 中国海洋大学 2024-05-28 CN disclosed