SCHEMBL30934591

SCHEMBL30934591

[2H]c1nccc2cc(NC(=O)[C@H](CNC(=O)OC(C)(C)C)c3ccc(COC(=O)c4ccc(C)cc4C)cc3)ccc12

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 17/20 0.65
ROCK1 Q13464 8/20 0.65
MYLK4 Q86YV6 1/20 0.48
TNF P01375 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23066372 1.00 ROCK2 (0.65) ROCK2ROCK1MYLK4TNF
SCHEMBL173486 0.93 ROCK2 (0.75) ROCK2ROCK1MYLK4TNF
SCHEMBL174353 0.93 ROCK2 (0.75) ROCK2ROCK1MYLK4TNF
SCHEMBL112454 0.93 ROCK2 (0.75) ROCK2ROCK1MYLK4TNF
SCHEMBL23066423 0.87 ROCK2 (0.65) ROCK2ROCK1MYLK4
Netarsudil SCHEMBL30934339 0.86 ROCK2 (0.85) ROCK2ROCK1MYLK4
Netarsudil SCHEMBL23066367 0.86 ROCK2 (0.85) ROCK2ROCK1MYLK4
Netarsudil SCHEMBL23066391 0.86 ROCK2 (0.76) ROCK2ROCK1MYLK4
SCHEMBL18827679 0.86 ROCK2 (0.73) ROCK2ROCK1MYLK4TNF
Netarsudil SCHEMBL23066437 0.85 ROCK2 (0.76) ROCK2ROCK1MYLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3768661-B1 DEUTERATED COMPOUNDS AS ROCK INHIBITORS FOCHON PHARMACEUTICALS LTD (CN) 2024-05-01 EP disclosed