SCHEMBL30944342

SCHEMBL30944342

CC1CCCC(C(=O)Nc2nc3ccccc3s2)C1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.57
RAB9A P51151 8/20 0.57
SMN1; SMN2 Q16637 6/20 0.57
ALDH1A1 P00352 4/20 0.57
TP53 P04637 2/20 0.57
MAPK1 P28482 1/20 0.57
ADORA1 P30542 1/20 0.56
DYRK1A Q13627 1/20 0.56
CYP1A2 P05177 1/20 0.55
GAA P10253 1/20 0.55
CYP2C19 P33261 1/20 0.55
MEN1 O00255 5/20 0.55
KMT2A Q03164 5/20 0.55
NFKB1 P19838 2/20 0.55
NFKB2 Q00653 2/20 0.55
RELA Q04206 2/20 0.55
KDM4E B2RXH2 2/20 0.54
CNR1 P21554 1/20 0.52
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6227837 0.88 GAA (0.68) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL4909101 0.84 NPC1 (0.70) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL30944345 0.84 CASP3 (0.72) NPC1RAB9ASMN1; SMN2ALDH1A1DYRK1A
SCHEMBL30944333 0.84 NPC1 (0.60) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL880500 0.83 GAA (0.76) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL30944360 0.82 NPC1 (0.61) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL30944319 0.82 KMT2A (0.61) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL28523859 0.82 NPC1 (0.61) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL30944344 0.82 ITK (0.64) NPC1RAB9ASMN1; SMN2ALDH1A1MAPK1
SCHEMBL30944364 0.81 CYP2D6 (0.80) NPC1RAB9ASMN1; SMN2ALDH1A1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN claimed
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN disclosed
CN-112423746-B Novel antimycobacterial heterocyclic amides 克莱斯通公司 2024-06-28 CN disclosed