SCHEMBL30944353

SCHEMBL30944353

O=C(Nc1nc2ccc(Cl)cc2s1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.70
CASP3 P42574 8/20 0.62
SENP8 Q96LD8 8/20 0.62
SENP7 Q9BQF6 8/20 0.62
SENP6 Q9GZR1 8/20 0.62
DYRK1A Q13627 1/20 0.60
FSCN1 Q16658 1/20 0.60
CYP2D6 P10635 1/20 0.59
CYP2B6 P20813 1/20 0.59
CYP2C19 P33261 1/20 0.59
NPC1 O15118 5/20 0.56
RAB9A P51151 5/20 0.56
SMN1; SMN2 Q16637 3/20 0.55
CLK1 P49759 3/20 0.55
ALDH1A1 P00352 1/20 0.55
MEN1 O00255 2/20 0.53
POLB P06746 2/20 0.53
KMT2A Q03164 2/20 0.53
HSD17B10 Q99714 1/20 0.53
KDM4E B2RXH2 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28529053 1.00 CNR1 (0.70) CNR1CASP3SENP8SENP7SENP6
SCHEMBL13778842 0.87 CNR1 (0.72) CNR1NPC1RAB9ASMN1; SMN2CLK1
SCHEMBL30944383 0.85 DYRK1A (0.56) CNR1CASP3SENP8SENP7SENP6
SCHEMBL4920969 0.83 NPC1 (0.75) CNR1DYRK1ACYP2C19NPC1RAB9A
SCHEMBL4918014 0.83 CNR1 (1.00) CNR1DYRK1ANPC1RAB9ASMN1; SMN2
SCHEMBL28512789 0.82 DYRK1A (0.58) CASP3SENP8SENP7SENP6DYRK1A
SCHEMBL30944286 0.82 DYRK1A (0.58) CASP3SENP8SENP7SENP6DYRK1A
SCHEMBL963747 0.82 CLK1 (0.76) CNR1NPC1RAB9ASMN1; SMN2CLK1
SCHEMBL30944323 0.81 CNR1 (0.64) CNR1DYRK1ACYP2C19NPC1RAB9A
SCHEMBL28527319 0.81 CNR1 (0.64) CNR1DYRK1ACYP2C19NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN claimed
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN disclosed
CN-112423746-B Novel antimycobacterial heterocyclic amides 克莱斯通公司 2024-06-28 CN disclosed