SCHEMBL30944944

SCHEMBL30944944

COc1ccc2nc(Nc3ccc(N4CCNCC4)cc3)cc(C(F)(F)F)c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 2/20 0.52
DNMT1 P26358 1/20 0.52
MAPT P10636 2/20 0.51
POLB P06746 2/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
KMT2A Q03164 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
HSD17B10 Q99714 1/20 0.51
KDM1A O60341 3/20 0.48
ADRB1 P08588 2/20 0.46
HTR3E A5X5Y0 1/20 0.46
HTR3B O95264 1/20 0.46
HTR3A P46098 1/20 0.46
HTR3D Q70Z44 1/20 0.46
HTR3C Q8WXA8 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
HTR1A P08908 1/20 0.46
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29230134 1.00 RAD52 (0.52) RAD52DNMT1MAPTPOLBTSHR
SCHEMBL30944974 0.89 DNMT1 (0.66) RAD52DNMT1MAPTPOLBTSHR
SCHEMBL29230399 0.89 DNMT1 (0.66) RAD52DNMT1MAPTPOLBTSHR
SCHEMBL29230140 0.85 KDM1A (0.47) KDM1ACDK4CCND1CCND2CCND3
SCHEMBL30944961 0.84 POLB (0.56) RAD52MAPTPOLBKMT2ASMN1; SMN2
SCHEMBL29230157 0.84 POLB (0.56) RAD52MAPTPOLBKMT2ASMN1; SMN2
SCHEMBL29230160 0.83 KDM1A (0.62) KDM1ASIGMAR1HTR1DCDK4CCND1
SCHEMBL30944977 0.83 ITGB3 (0.47) MAPTKMT2AKDM1ACDK4CCND1
SCHEMBL29230159 0.83 ITGB3 (0.47) MAPTKMT2AKDM1ACDK4CCND1
SCHEMBL30945029 0.82 GALR2 (0.50) RAD52DNMT1MAPTPOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118146151-A 4-Trifluoromethyl substituted quinoline and quinazoline compound and application thereof 贵州省中国科学院天然产物化学重点实验室(贵州医科大学天然产物化学重点实验室) 2024-06-07 CN disclosed